One-step synthesis of novel glycosyltransferase inhibitors.
نویسندگان
چکیده
A one-step synthesis of two 5-CF(3) UDP-sugars is reported. These non-natural sugar-nucleotides are micromolar inhibitors of two different galactosyltransferases.
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عنوان ژورنال:
- Chemical communications
دوره 48 97 شماره
صفحات -
تاریخ انتشار 2012